Stabilised GHRH analogue — human GHRH(1-44) amide, N-terminally acylated
Tesamorelin
An approved GHRH analogue and the only GHRH analogue in this library with a currently marketed United States approval.
Also listed as: Egrifta, TH9507, Tesamorelin acetate
Chemical identity
- Compound class
- Stabilised GHRH analogue — human GHRH(1-44) amide, N-terminally acylated
- Sequence
- trans-3-hexenoyl-GHRH(1-44)-NH2
- Molecular formula
- C221H366N72O67S
- Molecular weight
- 5136 g/mol
- CAS number
- 218949-48-5
- PubChem CID
- 16137828
- Research categories
- GHRH analogues, Approved drug substances
United States regulatory status
FDA-approved drug substance
BLA 022505 (EGRIFTA)
Marketed in the United States as EGRIFTA, an approved prescription product administered subcutaneously.
- EGRIFTA, BLA 022505, approved 10 November 2010. Active prescription product.
- Not listed on FDA's Category 2 or withdrawn-nomination compounding tables.
Anti-doping status
Named at S2.2.4 among GHRH analogues. Prohibited at all times; non-Specified.
Regulatory status describes how a substance is classified. It is not a safety assessment, and it says nothing about the quality of any particular material.
Evidence overview
3 records in this file
- CLINICAL TRIAL1
- REGULATORY2
Research areas. Anti-doping; Approved-drug Phase 3; United States approval.
Publication span. 2007–2026.
Open the evidence fileWhat we know
- FDA-approved as EGRIFTA (BLA 022505, 2010). Falutz et al. 2007 (NEJM) is a primary interventional paper in the HIV-lipodystrophy programme.
- It is the only GHRH analogue in this library with a currently marketed United States approval.
- Also named on the WADA GHRH-analogue list — approval and sporting prohibition are different questions.
Editorial reading of the records below, labelled as Therapept analysis. How records are built
What remains uncertain
- Orthopaedic or “performance” endpoints: 2026 sports-medicine reviews report no supporting evidence in those settings.
Sources
- PubChem CID 16137828
- Drugs@FDA — approved drug products
- WADA 2026 Prohibited ListEffective 1 January 2026.
Last reviewed 3 September 2026 · Compiled by Therapept Editorial · How these records are built
